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1 Ergebnisse
1
Structural and Activity Relationships of 6‑Sulfonyl-8-Nitro..:
Dongguang Fan (11525027)
;
Bin Wang (30851)
;
Giovanni Stelitano (6487385)
...
https://figshare.com/articles/journal_contribution/Structural_and_Activity_Relationships_of_6_Sulfonyl-8-Nitrobenzothiazinones_as_Antitubercular_Agents/16745969. , 1753
Link:
https://doi.org/10.1021/acs.jmedchem.1c01049.s001
RT Journal T1
Structural and Activity Relationships of 6‑Sulfonyl-8-Nitrobenzothiazinones as Antitubercular Agents
UL https://suche.suub.uni-bremen.de/peid=base-ftsmithonian:oai:figshare.com:article_16745969&Exemplar=1&LAN=DE A1 Dongguang Fan (11525027) A1 Bin Wang (30851) A1 Giovanni Stelitano (6487385) A1 Karin Savková (7297007) A1 Rui Shi (45165) A1 Stanislav Huszár (1667152) A1 Quanquan Han (11525030) A1 Katarína Mikušová (1446046) A1 Laurent R. Chiarelli (237358) A1 Yu Lu (11575) A1 Chunhua Qiao (544492) YR 1753 K1 Biochemistry K1 Medicine K1 Pharmacology K1 Biotechnology K1 Infectious Diseases K1 Environmental Sciences not elsewhere classified K1 Biological Sciences not elsewhere classified K1 Chemical Sciences not elsewhere classified K1 minimum inhibitory concentration K1 member aromatic heterocycles K1 low aqueous solubility K1 human liver microsomes K1 exploration introduced five K1 essential flavoenzyme dpre1 K1 bioavailability issues need K1 6 ‑ sulfonyl K1 38 </ b K1 exhibited mic 47 K1 6 </ b K1 potent antitubercular activity K1 btz derived compounds K1 extraordinarily potent K1 antitubercular agents K1 activity relationships K1 optimized compounds K1 based compounds K1 work led K1 study suggested K1 side chain K1 higher stability K1 druglike properties K1 consequently blocking K1 aryl group K1 alternative side K1 30 nm K1 2 ng JF https://figshare.com/articles/journal_contribution/Structural_and_Activity_Relationships_of_6_Sulfonyl-8-Nitrobenzothiazinones_as_Antitubercular_Agents/16745969 LK http://dx.doi.org/https://doi.org/10.1021/acs.jmedchem.1c01049.s001 DO https://doi.org/10.1021/acs.jmedchem.1c01049.s001 SF ELIB - SuUB Bremen
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