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1 Ergebnisse
1
Discovery of 2‑(Ortho-Substituted Benzyl)-Indole Derivative..:
Biao Lu (1342371)
;
Dong Liu (115204)
;
Bin Gui (542725)
...
https://figshare.com/articles/dataset/Discovery_of_2_Ortho-Substituted_Benzyl_-Indole_Derivatives_as_Potent_and_Orally_Bioavailable_ROR_Agonists_with_Antitumor_Activity/16803750. , 2021
Link:
https://doi.org/10.1021/acs.jmedchem.1c00828.s002
RT Journal T1
Discovery of 2‑(Ortho-Substituted Benzyl)-Indole Derivatives as Potent and Orally Bioavailable RORγ Agonists with Antitumor Activity
UL https://suche.suub.uni-bremen.de/peid=base-ftsmithonian:oai:figshare.com:article_16803750&Exemplar=1&LAN=DE A1 Biao Lu (1342371) A1 Dong Liu (115204) A1 Bin Gui (542725) A1 Jun Gou (2631100) A1 Huaide Dong (11558667) A1 Qiyue Hu (1963867) A1 Jun Feng (116162) A1 Yuchang Mao (11558670) A1 Xiaodong Shen (1542499) A1 Shenglan Wang (9611464) A1 Caihua Zhang (1802497) A1 Ru Shen (1758649) A1 Yinfa Yan (3005082) A1 Lei Chen (54296) A1 Huiyun Wang (3711682) A1 Di Li (335947) A1 Jiayin Zhang (1850089) A1 Minsheng Zhang (2403979) A1 Rumin Zhang (2729599) A1 Chang Bai (2356918) A1 Feng He (47348) A1 Weikang Tao (2428648) A1 Suxing Liu (1427581) YR 2021 K1 Biochemistry K1 Molecular Biology K1 Pharmacology K1 Biotechnology K1 Immunology K1 Cancer K1 Science Policy K1 Biological Sciences not elsewhere classified K1 Chemical Sciences not elsewhere classified K1 subtle structural differences K1 scaffold hopping based K1 functional drug target K1 first comprehensive work K1 activating anticancer agent K1 2 ‑( ortho K1 elicit antitumor efficacy K1 opposite biological moa K1 antitumor activity rorγ K1 17 </ b K1 antitumor efficacy K1 vivo </ K1 rorγ agonist K1 tumor tissues K1 rational optimization K1 pharmacokinetic profile K1 novel mechanism K1 compounds led K1 cancer immunity K1 also promotion JF https://figshare.com/articles/dataset/Discovery_of_2_Ortho-Substituted_Benzyl_-Indole_Derivatives_as_Potent_and_Orally_Bioavailable_ROR_Agonists_with_Antitumor_Activity/16803750 LK http://dx.doi.org/https://doi.org/10.1021/acs.jmedchem.1c00828.s002 DO https://doi.org/10.1021/acs.jmedchem.1c00828.s002 SF ELIB - SuUB Bremen
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