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1 Ergebnisse
1
N‑Terminus to Arginine Side-Chain Cyclization of Linear Pep..:
Adam Konieczny (7461407)
;
Marcus Conrad (272293)
;
Fabian J. Ertl (11662728)
...
https://figshare.com/articles/journal_contribution/N_Terminus_to_Arginine_Side-Chain_Cyclization_of_Linear_Peptidic_Neuropeptide_Y_Y_sub_4_sub_Receptor_Ligands_Results_in_Picomolar_Binding_Constants/16955766. , 2021
Link:
https://doi.org/10.1021/acs.jmedchem.1c01574.s003
RT Journal T1
N‑Terminus to Arginine Side-Chain Cyclization of Linear Peptidic Neuropeptide Y Y 4 Receptor Ligands Results in Picomolar Binding Constants
UL https://suche.suub.uni-bremen.de/peid=base-ftsmithonian:oai:figshare.com:article_16955766&Exemplar=1&LAN=DE A1 Adam Konieczny (7461407) A1 Marcus Conrad (272293) A1 Fabian J. Ertl (11662728) A1 Jakob Gleixner (11662731) A1 Albert O. Gattor (11662734) A1 Lukas Grätz (8855417) A1 Maximilian F. Schmidt (6693701) A1 Eduard Neu (11662737) A1 Anselm H. C. Horn (11662740) A1 David Wifling (453030) A1 Peter Gmeiner (217594) A1 Timothy Clark (425636) A1 Heinrich Sticht (173676) A1 Max Keller (113018) YR 2021 K1 Biophysics K1 Biochemistry K1 Molecular Biology K1 Pharmacology K1 Biotechnology K1 Hematology K1 Biological Sciences not elsewhere classified K1 Chemical Sciences not elsewhere classified K1 represent promising leads K1 picomolar binding constants K1 e K1 n K1 receptor ligands results K1 linear precursor peptides K1 5 </ sub K1 4 </ sub K1 2 </ sub K1 1 </ sub K1 r partial agonists K1 n ‑ terminus K1 linear peptidic neuropeptide K1 labeled tool compounds K1 human pancreatic polypeptide K1 npy K1 2 +</ sup K1 18 </ b K1 r affinity compared K1 </ sub K1 pancreatic polypeptide K1 k </ K1 r ligands K1 r affinity K1 peptides acted K1 >< sub K1 r selectivity K1 r potency K1 r ) K1 peptide yy K1 novel approach K1 might support K1 hpp ) K1 fold higher K1 cyclic oligopeptidic K1 chain cyclization K1 arginine side K1 also higher K1 aequorin assay JF https://figshare.com/articles/journal_contribution/N_Terminus_to_Arginine_Side-Chain_Cyclization_of_Linear_Peptidic_Neuropeptide_Y_Y_sub_4_sub_Receptor_Ligands_Results_in_Picomolar_Binding_Constants/16955766 LK http://dx.doi.org/https://doi.org/10.1021/acs.jmedchem.1c01574.s003 DO https://doi.org/10.1021/acs.jmedchem.1c01574.s003 SF ELIB - SuUB Bremen
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