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Into Deep Water: Optimizing BCL6 Inhibitors by Growing into..:
Matthew G. Lloyd (1804930)
;
Rosemary Huckvale (6734207)
;
Kwai-Ming J. Cheung (1266996)
...
https://figshare.com/articles/journal_contribution/Into_Deep_Water_Optimizing_BCL6_Inhibitors_by_Growing_into_a_Solvated_Pocket/17102290. , 2021
Link:
https://doi.org/10.1021/acs.jmedchem.1c00946.s002
RT Journal T1
Into Deep Water: Optimizing BCL6 Inhibitors by Growing into a Solvated Pocket
UL https://suche.suub.uni-bremen.de/peid=base-ftsmithonian:oai:figshare.com:article_17102290&Exemplar=1&LAN=DE A1 Matthew G. Lloyd (1804930) A1 Rosemary Huckvale (6734207) A1 Kwai-Ming J. Cheung (1266996) A1 Matthew J. Rodrigues (8697474) A1 Gavin W. Collie (1970749) A1 Olivier A. Pierrat (1276839) A1 Mahad Gatti Iou (9212736) A1 Michael Carter (3480731) A1 Owen A. Davis (1336125) A1 P. Craig McAndrew (4740555) A1 Emma Gunnell (11773213) A1 Yann-Vaï Le Bihan (8697486) A1 Rachel Talbot (4012325) A1 Alan T. Henley (1353570) A1 Louise D. Johnson (8697480) A1 Angela Hayes (1282245) A1 Michael D. Bright (8697471) A1 Florence I. Raynaud (1269372) A1 Mirco Meniconi (11773216) A1 Rosemary Burke (185752) A1 Rob L. M. van Montfort (8697498) A1 Olivia W. Rossanese (1352277) A1 Benjamin R. Bellenie (2712163) A1 Swen Hoelder (421014) YR 2021 K1 Biochemistry K1 Pharmacology K1 Immunology K1 Inorganic Chemistry K1 Hematology K1 Biological Sciences not elsewhere classified K1 Chemical Sciences not elsewhere classified K1 Physical Sciences not elsewhere classified K1 Information Systems not elsewhere classified K1 forming new interactions K1 formed hydrogen bonds K1 filled protein pockets K1 finding productive ways K1 25 </ b K1 optimizing bcl6 inhibitors K1 potent inhibitors K1 work highlights K1 ultimately achieving K1 systematically probing K1 submicromolar inhibition K1 sequential manner K1 satisfactory pharmacokinetic K1 remaining two K1 promising profile K1 increasing fashion K1 fold improvement K1 deep water K1 also perturbing JF https://figshare.com/articles/journal_contribution/Into_Deep_Water_Optimizing_BCL6_Inhibitors_by_Growing_into_a_Solvated_Pocket/17102290 LK http://dx.doi.org/https://doi.org/10.1021/acs.jmedchem.1c00946.s002 DO https://doi.org/10.1021/acs.jmedchem.1c00946.s002 SF ELIB - SuUB Bremen
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