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1 Ergebnisse
1
Discovery of Spiro-azaindoline Inhibitors of Hematopoietic ..:
Bryan K. Chan (1346358)
;
Eileen Seward (1436785)
;
Michael Lainchbury (1290594)
...
https://figshare.com/articles/journal_contribution/Discovery_of_Spiro-azaindoline_Inhibitors_of_Hematopoietic_Progenitor_Kinase_1_HPK1_/17144017. , 2021
Link:
https://doi.org/10.1021/acsmedchemlett.1c00473.s001
RT Journal T1
Discovery of Spiro-azaindoline Inhibitors of Hematopoietic Progenitor Kinase 1 (HPK1)
UL https://suche.suub.uni-bremen.de/peid=base-ftsmithonian:oai:figshare.com:article_17144017&Exemplar=1&LAN=DE A1 Bryan K. Chan (1346358) A1 Eileen Seward (1436785) A1 Michael Lainchbury (1290594) A1 Thomas F. Brewer (1321218) A1 Le An (4453327) A1 Toby Blench (2316310) A1 Matthew W. Cartwright (2069500) A1 Grace Ka Yan Chan (11705515) A1 Edna F. Choo (1728364) A1 Jason Drummond (1845673) A1 Richard L. Elliott (2119969) A1 Emanuela Gancia (1577419) A1 Lewis Gazzard (1464970) A1 Baihua Hu (1600627) A1 Graham E. Jones (11811712) A1 Xifeng Luo (2553394) A1 Andrew Madin (2369338) A1 Sushant Malhotra (1784344) A1 John G. Moffat (413533) A1 Jodie Pang (1429792) A1 Laurent Salphati (1443862) A1 Christopher J. Sneeringer (10493104) A1 Craig E. Stivala (1861234) A1 Binqing Wei (2069518) A1 Weiru Wang (640332) A1 Ping Wu (46628) A1 Timothy P. Heffron (1346370) YR 2021 K1 Biochemistry K1 Cell Biology K1 Genetics K1 Molecular Biology K1 Physiology K1 Pharmacology K1 Biotechnology K1 Immunology K1 Cancer K1 Hematology K1 Infectious Diseases K1 Virology K1 Computational Biology K1 Biological Sciences not elsewhere classified K1 Chemical Sciences not elsewhere classified K1 tumor growth inhibition K1 throughput screening hit K1 induce cytokine production K1 small molecule inhibitors K1 azaindoline inhibitors K1 vitro </ K1 unusual p K1 significantly improved K1 primary human K1 physicochemical property K1 negative regulator K1 metabolic liabilities K1 kinase selectivity K1 initial 7 K1 glioma models K1 dead knock K1 cell receptor K1 cell function K1 cell activation K1 based optimization K1 azaindole high K1 adme properties JF https://figshare.com/articles/journal_contribution/Discovery_of_Spiro-azaindoline_Inhibitors_of_Hematopoietic_Progenitor_Kinase_1_HPK1_/17144017 LK http://dx.doi.org/https://doi.org/10.1021/acsmedchemlett.1c00473.s001 DO https://doi.org/10.1021/acsmedchemlett.1c00473.s001 SF ELIB - SuUB Bremen
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