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1 Ergebnisse
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Lead optimization of a pyrazolo[1,5-a]pyrimidin-7(4H)-one s..:
Liang, Jun
;
Zhang, Birong
;
Labadie, Sharada
...
Bioorganic & Medicinal Chemistry Letters. 26 (2016) 16 - p. 4036-4041 , 2016
Link:
https://doi.org/10.1016/j.bmcl.2016.06.078
RT Journal T1
Lead optimization of a pyrazolo[1,5-a]pyrimidin-7(4H)-one scaffold to identify potent, selective and orally bioavailable KDM5 inhibitors suitable for in vivo biological studies
UL https://suche.suub.uni-bremen.de/peid=cr-10.1016_j.bmcl.2016.06.078&Exemplar=1&LAN=DE A1 Liang, Jun A1 Zhang, Birong A1 Labadie, Sharada A1 Ortwine, Daniel F. A1 Vinogradova, Maia A1 Kiefer, James R. A1 Gehling, Victor S. A1 Harmange, Jean-Christophe A1 Cummings, Richard A1 Lai, Tommy A1 Liao, Jiangpeng A1 Zheng, Xiaoping A1 Liu, Yichin A1 Gustafson, Amy A1 Van der Porten, Erica A1 Mao, Weifeng A1 Liederer, Bianca M. A1 Deshmukh, Gauri A1 Classon, Marie A1 Trojer, Patrick A1 Dragovich, Peter S. A1 Murray, Lesley PB Elsevier BV YR 2016 SN 0960-894X JF Bioorganic & Medicinal Chemistry Letters VO 26 IS 16 SP 4036 OP 4041 LK http://dx.doi.org/https://doi.org/10.1016/j.bmcl.2016.06.078 DO https://doi.org/10.1016/j.bmcl.2016.06.078 SF ELIB - SuUB Bremen
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